Acetaldehyde → HCID 54121951, compound

Participants

Reaction Steps

4-Amino-5-chloro-N-((1-(5-(3,4-dichlorobenzylamino)pentyl)-piperidin-4-yl)methyl)-2-methoxybenzamide (2.0 g) as starting compound, acetaldehyde (0.27 ml) and sodium cyanoborohydride (0.3 g) were reacted and treated in the same manner as in Example 136 to give 0.82 g of 4-amino-5-chloro-N-((1-(5-(N-(3,4-dichlorobenzyl)-N-ethylamino)pentyl)-piperidin-4-yl)methyl)-2-methoxybenzamide.

Provenance & Evidence