Acetaldehyde → HCID 54317976, compound

Participants

Reaction Steps

4-Amino-5-chloro-N-((1-(4-(3,4-dichlorobenzylamino)butyl)piperidin-4-yl)methyl)-2-methoxybenzamide (1.9 g) as starting compound, acetaldehyde (0.26 ml) and sodium cyanoborohydride (0.3 g) were reacted and treated in the same manner as in Example 136 to give 1.1 g of 4-amino-5-chloro-N-((1-(4-(N-(3,4-dichlorobenzyl)-N-ethylamino)butyl)-piperidin-4-yl)methyl)-2-methoxybenzamide.

Provenance & Evidence