反应详情

Following the general procedure of EXAMPLE 70, and making non-critical variations but substituting 1-benzyl-4-(1-cyclopentylamino)piperidine (EXAMPLE 103) for 1-benzyl-4-(methylamino)piperidine and 2-chloro-3-nitropyridine for 2-bromo-3-ethoxypyridine and using a reaction time of 2 hrs, the title compound is obtained, NMR (CDCl3) 8.26, 7.91, 7.33-7.21, 6.67, 3.78, 3.47, 2.97-2.86, 2.11, 1.98-1.75 and 1.50δ.

1. customa reaction time of 2 hrs