HCID 20352979, compound → HCID 20352934, compound
Reaction equation
CN[CH:3]([C:6]1C=C[CH:9]=[CH:8][C:7]=1C)[CH2:4]N.[CH2:13]([N:15]1[CH:19]([C:20]2[CH:25]=[CH:24][CH:23]=[CH:22][CH:21]=2)[CH2:18][N:17]=[C:16]1[NH:26][C:27]([O:29][CH3:30])=[O:28])C>>[CH3:13][N:15]1[CH:19]([C:20]2[CH:25]=[CH:24][C:23]([CH2:4][CH2:3][CH2:6][CH2:7][CH2:8][CH3:9])=[CH:22][CH:21]=2)[CH2:18][N:17]=[C:16]1[NH:26][C:27]([O:29][CH3:30])=[O:28]Participants
Procedure
Similarly, by following the same procedure of part A but respectively replacing the β-methylamino-β-(2-methylphenyl)-ethylamine with other β-alkylamino-β-phenylethylamino or β-alkylamino-(substituted phenyl)-ethylamino such as β-ethylamino-β-phenylethylamine β-isopropylamino-β-(substituted phenyl)-ethylamine, β-t-butylamino-β-(substituted phenyl)-ethylamine, β-isoamylamino-β-(substituted phenyl)-ethylamine, β-2'-t-butylethylamino-β-(substituted phenyl)-ethylamine, or β-n-hexylamino-β-(substituted phenyl)-ethylamine, the corresponding 1-alkyl-4,5-dihydro-5-(substituted phenyl)-2-methoxycarbonylaminoimidazole or 1-alkyl-4,5-dihydro-5-phenyl-2-methoxycarbonylaminoimidazoles such as 1-ethyl-4,5-dihydro-5-phenyl-2-methoxycarbonylaminoimidazole, m.p. 115°-116° C;
Sources & evidence
- ORD record
- ord-80a96ff999d14a16af3d907760b5b305
- Source dataset
- uspto-grants-1978_05
- Patent number
- US04088771
Reaction notes
Loading…