Phenylmethanesulfonyl chloride → [4-Chloro-2-[[2-methyl-4-[(phenylmethyl)sulfonyl]-1-piperazinyl]methyl]phenoxy]acetic acid

HRID 38266Notes

Reaction equation

HRID 38266 reaction equation
[Cl:1][C:2]1[CH:12]=[CH:11][C:5]([O:6][CH2:7][C:8]([OH:10])=[O:9])=[C:4]([CH2:13][N:14]2[CH2:19][CH2:18][N:17]([S:20]([C:23]3[CH:28]=[CH:27][CH:26]=[CH:25][CH:24]=3)(=[O:22])=[O:21])[CH2:16][CH:15]2[CH3:29])[CH:3]=1.[CH:30]1C=CC(CS(Cl)(=O)=O)=CC=1>>[Cl:1][C:2]1[CH:12]=[CH:11][C:5]([O:6][CH2:7][C:8]([OH:10])=[O:9])=[C:4]([CH2:13][N:14]2[CH2:19][CH2:18][N:17]([S:20]([CH2:23][C:24]3[CH:30]=[CH:28][CH:27]=[CH:26][CH:25]=3)(=[O:21])=[O:22])[CH2:16][CH:15]2[CH3:29])[CH:3]=1

Participants

3

Procedure

Prepared by the method of example 30, using the product of example 53 part (b) and benzenemethanesulfonyl chloride to give the title compound.

Workup

  1. customPrepared by the method of example 30

Sources & evidence

ORD record
ord-4ce17325f6504feaab3e708fcc28b51d
Source dataset
uspto-grants-2013_09
Patent number
US08524715B2

Reaction notes

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