Benzenesulfonyl chloride → [4-Chloro-2-[[3-methyl-4-(phenylsulfonyl)-1-piperazinyl]methyl]phenoxy]acetic Acid

HRID 38267Notes

Reaction equation

HRID 38267 reaction equation
[Cl:1][C:2]1[CH:12]=[CH:11][C:5]([O:6][CH2:7][C:8]([OH:10])=[O:9])=[C:4]([CH2:13][N:14]2[CH2:19][CH2:18][N:17]([S:20]([CH2:23][C:24]3[CH:29]=[CH:28][CH:27]=[CH:26]C=3)(=[O:22])=[O:21])[CH:16]([CH3:30])[CH2:15]2)[CH:3]=1.C1(S(Cl)(=O)=O)C=CC=CC=1>>[Cl:1][C:2]1[CH:12]=[CH:11][C:5]([O:6][CH2:7][C:8]([OH:10])=[O:9])=[C:4]([CH2:13][N:14]2[CH2:19][CH2:18][N:17]([S:20]([C:23]3[CH:26]=[CH:27][CH:28]=[CH:29][CH:24]=3)(=[O:21])=[O:22])[CH:16]([CH3:30])[CH2:15]2)[CH:3]=1

Participants

3

Procedure

Prepared by the method of example 30, using the product from example 56 part (a) and is benzenesulfonyl chloride to give the title compound.

Workup

  1. customPrepared by the method of example 30

Sources & evidence

ORD record
ord-a876609625a94e64a22f39f164b58057
Source dataset
uspto-grants-2013_09
Patent number
US08524715B2

Reaction notes

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