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HuagongsheHuagongshe Chemistry Print Report · For research reference only
HRID 383296Generated: October 29, 2026

(3-(1H-pyrazol-1-yl)phenyl)boronic acid → (1RS,3RS)-3-[3-(3-Pyrazol-1-yl-phenyl)-imidazo[1,2-a]pyridin-6-ylamino]-cyclohexanol

https://huagongshe.com/reaction/383296

Reaction equation

Participants

RoleNameHCIDCharge
Reactant(3-(1H-pyrazol-1-yl)phenyl)boronic acidHCID 16640530—
Reactant(1RS,3RS)-3-(3-Bromo-imidazo[1,2-a]pyridin-6-ylamino)-cyclohexanolHCID 68483082—
Product(1RS,3RS)-3-[3-(3-Pyrazol-1-yl-phenyl)-imidazo[1,2-a]pyridin-6-ylamino]-cyclohexanolHCID 68487287—

Reaction Steps

This compound is prepared from (1RS,3RS)-3-(3-Bromo-imidazo[1,2-a]pyridin-6-ylamino)-cyclohexanol (Intermediate J [step 1]) and 3-(1H-pyrazol-1-yl)-phenylboronic acid analogously to Example 2.1 (step 2)

Provenance & Evidence

DOI10.6084/m9.figshare.5104873.v1
Patent numberUS08367662B2
Source datasetuspto-grants-2013_02
ORD IDord-ee0a3421f5644f83b284efcab23307a1
Source noteuspto-grants-2013_02