Potassium Carbonate → 3-amino-1-{(4-phenylpiperazin-1-yl)propanoyl}-6-N-(p-tolyl)-4,5,6,7-tetrahydro-1H-pyrazolo[3,4-c]pyridin-7-one

Participants

Reaction Steps

A target compound (77.8 mg, 0.169 mmol, 44.7%) was yielded as liquid in the same manner as Example 1 by reacting 1-N-t-butoxycarbonyl-3-amino-4,5,6,7-tetrahydro-6-N-(p-tolyl)pyrazolo[3,4-c]pyridin-7-one (130 mg, 0.379 mmol) with potassium carbonate (57.6 mg, 0.417 mmol) and 3-chloro-1-(4-phenylpiperazin-1-yl)propan-1-one (100.6 mg, 0.398 mmol).

Provenance & Evidence