Potassium Carbonate → 3-amino-1-[{4-(2,4,5-trimethylphenyl)piperazin-1-yl}propanoyl]-6-N-(p-tolyl)-4,5,6,7-tetrahydro-1H-pyrazolo[3,4-c]pyridin-7-one

Participants

Reaction Steps

A target compound (107.5 mg, 0.214 mmol, 53.7%) was yielded as solid in the same manner as Example 1 by reacting 3-amino-5,6-dihydro-6-N-(p-tolyl)-1H-pyrazolo[3,4-c]pyridin-7(4H)-one (97 mg, 0.4 mmol) with potassium carbonate (82.9 mg, 0.6 mmol) and 3-chloro-1-{4-(2,4,5-trimethylphenyl)piperazin-1-yl}propan-1-one (129.7 mg, 0.44 mmol).

Provenance & Evidence