Triethylamine → HCID 178440409, compound

Participants

Reaction Steps

Analogously to the procedure of Example 5, starting from 34 mg (0.115 mmol) of 5-(4-amino-2,6-dimethylphenoxy)-3-propyl-1H-indazole, 11.6 mg (0.115 mmol) of triethylamine and 15.7 mg (0.115 mmol) of ethyl oxalyl chloride, 18 mg, (32%) of ethyl [5-(4-{[ethoxy(oxo)acetyl]amino}-2,6-dimethylphenoxy)-3-propyl-1H-indazol-1-yl](oxo)acetate (Example 8) are obtained. Moreover, 18 mg, (40%) of ethyl ({3,5-dimethyl-4-[(3-propyl-1H-indazol-5-yl)oxy]phenyl}amino)(oxo)acetate (Example 8a) are obtained.

Provenance & Evidence