3-Pyridinylboronic acid → HCID 23003470, compound

HRID 396527Notes

Reaction equation

HRID 396527 reaction equation
[CH3:1][O:2][C:3](=[O:24])[CH2:4][C:5]1[C:13]2[C:8](=[CH:9][C:10]([Cl:14])=[CH:11][CH:12]=2)[NH:7][C:6]=1[C:15](=[O:23])[C:16]1[CH:21]=[CH:20][C:19](Br)=[CH:18][CH:17]=1.[N:25]1[CH:30]=[CH:29][CH:28]=[C:27](B(O)O)[CH:26]=1>>[CH3:1][O:2][C:3](=[O:24])[CH2:4][C:5]1[C:13]2[C:8](=[CH:9][C:10]([Cl:14])=[CH:11][CH:12]=2)[NH:7][C:6]=1[C:15](=[O:23])[C:16]1[CH:21]=[CH:20][C:19]([C:27]2[CH:26]=[N:25][CH:30]=[CH:29][CH:28]=2)=[CH:18][CH:17]=1

Participants

3

Reactant 2

HCID 27343783-Pyridinylboronic acidHCID 23003358HCID 23003358, compound

Product 1

HCID 23003470HCID 23003470, compound

Procedure

The title compound was prepared according to the procedure described in Example 207 from methyl[6-chloro-2-(4-bromobenzoyl)-1H-indol-3-yl]acetate (Example 206) and pyridine-3-boronic acid.

Sources & evidence

ORD record
ord-068b454f13874b4b9baada7d72b93f40
Source dataset
uspto-grants-2003_08
Patent number
US06608070B1

Reaction notes

Loading…