(Pyrimidin-5-yl)boronic acid → HCID 86670610, compound

HRID 401462Notes

Reaction equation

HRID 401462 reaction equation
Br[C:2]1[CH:3]=[CH:4][C:5]2[N:6]([C:8]([CH:11]=[O:12])=[CH:9][N:10]=2)[CH:7]=1.[N:13]1[CH:18]=[C:17](B(O)O)[CH:16]=[N:15][CH:14]=1>>[N:13]1[CH:18]=[C:17]([C:2]2[CH:3]=[CH:4][C:5]3[N:6]([C:8]([CH:11]=[O:12])=[CH:9][N:10]=3)[CH:7]=2)[CH:16]=[N:15][CH:14]=1

Participants

3

Reactant 2

HCID 2795193(Pyrimidin-5-yl)boronic acidHCID 213456766-Bromoimidazo[1,2-a]pyridine-3-carbaldehyde2×

Product 1

HCID 86670610HCID 86670610, compoundYield 50%

Procedure

The title compound was prepared by following the procedure as described for Intermediate 1 using 6-bromoimidazo[1,2-a]pyridine-3-carbaldehyde and pyrimidin-5-ylboronic acid.

Sources & evidence

ORD record
ord-1d86a5511ce2466bbcaa4095f5e1beb3
Source dataset
uspto-grants-2014_06
Patent number
US08741932B2

Reaction notes

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