反应详情

As described for example 35b, 6-[5-(5-fluoro-pyridin-2-yl)-3-methyl-3H-[1,2,3]triazol-4-ylmethoxy]-nicotinic acid (80 mg, 0.24 mmol) was converted, using 4-aminomorpholine instead of 4-aminotetrahydropyran, to the title compound (87 mg, 87%) which was obtained as a white solid. MS: m/e=414.4 [M+H]+.