反应详情

As described for example 80c, 5-[3-(4-fluoro-phenyl)-5-methyl-3H-[1,2,3]triazol-4-ylmethoxy]-pyrazine-2-carboxylic acid (83 mg, 0.25 mmol), was converted, using 4-aminomorpholine instead of 4-aminotetrahydropyran, to the title compound (62 mg, 60%) which was obtained as a white solid. MS: m/e=414.4 [M+H]+.