4-Bromo-3-methylaniline → HCID 42637700, compound

HRID 405200Notes

Reaction equation

HRID 405200 reaction equation
[Cl:1][C:2]1[C:7]([Cl:8])=[CH:6][CH:5]=[CH:4][C:3]=1B(O)O.Br[C:13]1[CH:19]=[CH:18][C:16]([NH2:17])=[CH:15][C:14]=1C.ClC1C=CC(B(O)O)=CC=1>>[Cl:1][C:2]1[C:7]([Cl:8])=[CH:6][CH:5]=[CH:4][C:3]=1[C:13]1[CH:19]=[CH:18][C:16]([NH2:17])=[CH:15][CH:14]=1

Participants

4

Reactant 3

HCID 233594-Bromo-3-methylanilineHCID 742994-Chlorophenylboronic acidHCID 27346612,3-Dichlorobenzeneboronic acid

Product 1

HCID 42637700HCID 42637700, compound

Procedure

The title compound was prepared as described in Example 76, STEP B, substituting 4-iodoaniline and 2,3-dichlorophenylboronic acid for 4-bromo-3-methylaniline and 4-chlorophenylboronic acid.

Sources & evidence

ORD record
ord-e3a697d069f5428f971962c7ef2a3382
Source dataset
uspto-grants-2014_06
Patent number
US08748624B2

Reaction notes

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