4-Iodoanisole → 1-(4-methoxyphenyl)-1H-indazol-4-amine

HRID 418764Notes

Reaction equation

HRID 418764 reaction equation
F[C:2]1[CH:7]=[CH:6][CH:5]=[CH:4][C:3]=1[N:8]1[C:16]2[CH:15]=[CH:14][CH:13]=[C:12]([NH2:17])[C:11]=2[CH:10]=[N:9]1.N1C2C=CC=C(N)C=2C=N1.IC1C=C[C:32]([O:35]C)=CC=1>>[CH3:32][O:35][C:6]1[CH:5]=[CH:4][C:3]([N:8]2[C:16]3[CH:15]=[CH:14][CH:13]=[C:12]([NH2:17])[C:11]=3[CH:10]=[N:9]2)=[CH:2][CH:7]=1

Participants

4

Reactant 3

HCID 696764-IodoanisoleHCID 413085NoName_3327HCID 576159581-(2-Fluorophenyl)-1H-indazol-4-amine

Product 1

HCID 576159491-(4-methoxyphenyl)-1H-indazol-4-amine

Procedure

Similarly prepared to Intermediate 1 from 1H-indazol-4-amine and 1-iodo-4-(methyloxy)benzene.

Sources & evidence

ORD record
ord-9c811384d67f4e1fa44fd78594fd1e91
Source dataset
uspto-grants-2012_01
Patent number
US08093281B2

Reaction notes

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