Iodobenzene → 6-Methyl-1-phenyl-1H-indazol-4-amine

HRID 418770Notes

Reaction equation

HRID 418770 reaction equation
[NH2:1][C:2]1[CH:10]=[CH:9][CH:8]=[C:7]2[C:3]=1[CH:4]=[N:5][N:6]2[C:11]1[CH:12]=[C:13]([CH:18]=[CH:19][CH:20]=1)C(OC)=O.[CH3:21]C1C=C(N)C2C=NNC=2C=1.IC1C=CC=CC=1>>[CH3:21][C:9]1[CH:10]=[C:2]([NH2:1])[C:3]2[CH:4]=[N:5][N:6]([C:11]3[CH:20]=[CH:19][CH:18]=[CH:13][CH:12]=3)[C:7]=2[CH:8]=1

Participants

4

Reactant 3

HCID 11575IodobenzeneHCID 193544286-Methyl-1H-indazol-4-amineHCID 57615925Methyl 3-(4-amino-1H-indazol-1-yl)benzoate

Product 1

HCID 249380596-Methyl-1-phenyl-1H-indazol-4-amine

Procedure

Similarly prepared to Intermediate 9 from 6-methyl-1H-indazol-4-amine and iodobenzene.

Sources & evidence

ORD record
ord-13f9b8d113a34d4592a941452e293bd3
Source dataset
uspto-grants-2012_01
Patent number
US08093281B2

Reaction notes

Loading…