3-Fluorophenylboronic acid → HCID 59252462, compound

Participants

Reaction Steps

The title compound was prepared according to the method described in Example 22, except that (±)-tert-butyl 3-(4-(2-phenylpyrimidin-5-yl)-1H-imidazol-2-yl)pyrrolidine-1-carboxylate (Example 28) was used instead of (±)-tert-butyl 3-(4-(2-phenylpyrimidin-5-yl)-1H-imidazol-2-yl)piperidine-1-carboxylate. MS (ESI+) m/z 292 (M+1); H-PGDS FPBA IC50: 2 μM.

Provenance & Evidence