2-methyl-3-(1,2,3,6-tetrahydropyridin-4-yl)-1H-indole → HCID 9845207, compound

HRID 431635Notes

Reaction equation

HRID 431635 reaction equation
[CH3:1][N:2]([S:16]([C:19]1[CH:20]=[C:21]([CH3:25])[CH:22]=[CH:23][CH:24]=1)(=[O:18])=[O:17])[CH2:3][CH2:4]OS(C1C=C(C)C=CC=1)(=O)=O.[CH3:26][C:27]1[NH:28][C:29]2[C:34]([C:35]=1[C:36]1[CH2:37][CH2:38][NH:39][CH2:40][CH:41]=1)=[CH:33][CH:32]=[CH:31][CH:30]=2>>[CH3:25][C:21]1[CH:20]=[C:19]([S:16]([N:2]([CH3:1])[CH2:3][CH2:4][N:39]2[CH2:40][CH:41]=[C:36]([C:35]3[C:34]4[C:29](=[CH:30][CH:31]=[CH:32][CH:33]=4)[NH:28][C:27]=3[CH3:26])[CH2:37][CH2:38]2)(=[O:17])=[O:18])[CH:24]=[CH:23][CH:22]=1

Participants

3

Reactant 2

HCID 32454072-methyl-3-(1,2,3,6-tetrahydropyridin-4-yl)-1H-indoleHCID 11485905HCID 11485905, compound

Product 1

HCID 9845207HCID 9845207, compound

Procedure

The title compound was prepared using the procedure described in Example 1 using toluene-3-sulfonic acid 2-(methyl-(toluene-3-sulfonyl)-amino)-ethyl ester (D1) and 2-methyl-3-(1,2,3,6-tetrahydro-pyridin-4-yl)-1H indole. MH+ 424.

Sources & evidence

ORD record
ord-93713d97606c4787a3056ea74bfd8fda
Source dataset
uspto-grants-2003_12
Patent number
US06660751B1

Reaction notes

Loading…