HuagongsheHuagongshe Chemistry Print Report · For research reference only
(2S)-2-[[2-(3,5-difluorophenyl)acetyl]amino]propanoic acid → 3-(N'-(3,5-Difluorophenylacetyl)-L-alaninyl)amino-delta-valerolactam
Participants
| Role | Name | HCID | Charge |
|---|---|---|---|
| Reactant | (2S)-2-[[2-(3,5-difluorophenyl)acetyl]amino]propanoic acid | HCID 12135350 | — |
| Reactant | 4-Aminopiperidin-2-one | HCID 19980260 | — |
| Product | 3-(N'-(3,5-Difluorophenylacetyl)-L-alaninyl)amino-delta-valerolactam | HCID 9967722 | — |
Reaction Steps
Following General Procedure A and using N-(3,5-difluorophenylacetyl)-L-alanine (Example B) and 3-amino-δ-valerolactam (prepared by the procedure of D. W. Adamson, J. Chem. Soc. 1943, 39), the title compound was prepared.
Provenance & Evidence
| DOI | 10.6084/m9.figshare.5104873.v1 |
|---|---|
| Patent number | US06667305B1 |
| Source dataset | uspto-grants-2003_12 |
| ORD ID | ord-003fdae7255149d8b3059f770a1844f0 |
| Source note | uspto-grants-2003_12 |