HCID 178422395, compound → HCID 178503068, compound

HRID 441660Notes

Reaction equation

HRID 441660 reaction equation
[NH:1]1[C:5]([NH:6][C:7]([C:9]2[C:17](=[O:18])[N:16]3[C:12]([S:13][C:14]4[CH:22]=[C:21](C)[C:20]([NH2:24])=[CH:19][C:15]=43)=[N:11][CH:10]=2)=[O:8])=[N:4][N:3]=[N:2]1.N1C(NC(C2C(=O)N3[C:36]([S:37]C4C=C(CCC)C(N)=CC=43)=NC=2)=O)=NN=N1.N1C(NC(C2C(=O)N3C(SC4C=C(OC)C(N)=CC=43)=NC=2)=O)=NN=N1.N1C(NC(C2C(=O)N3C(SC4C=C(OCC)C(N)=CC=43)=NC=2)=O)=NN=N1.N1C(NC(C2C(=O)N3C(SC4C=C(O)C(N)=CC=43)=NC=2)=O)=NN=N1.N1C(NC(C2C(=O)N3C(SC4C=C(Cl)C(N)=CC=43)=NC=2)=O)=NN=N1.N1C(NC(C2C(=O)N3C(SC4C=C(F)C(N)=CC=43)=NC=2)=O)=NN=N1>>[NH:4]1[C:5]([NH:6][C:7]([C:9]2[C:17](=[O:18])[N:16]3[C:12]([S:13][C:14]4[CH:22]=[C:21]([S:37][CH3:36])[C:20]([NH2:24])=[CH:19][C:15]=43)=[N:11][CH:10]=2)=[O:8])=[N:1][N:2]=[N:3]1

Participants

8

Reactant 7

HCID 178422395HCID 178422395, compoundHCID 178438410HCID 178438410, compoundHCID 178465856HCID 178465856, compoundHCID 178486929HCID 178486929, compoundHCID 178507191HCID 178507191, compoundHCID 178507193HCID 178507193, compoundHCID 178507197HCID 178507197, compound

Product 1

HCID 178503068HCID 178503068, compound

Procedure

N-(5-tetrazolyl)-7-amino-8-methyl-4-oxo-4H-pyrimido[2,1-b]benzothiazole-3-carboxamide; N-(5-tetrazolyl)-7-amino-8-n-propyl-4-oxo-4H-pyrimido[2,1-b]benzothiazole-3-carboxamide; N-(5-tetrazolyl)-7-amino-8-methoxy-4-oxo-4H-pyrimido[2,1-b]benzothiazole-3-carboxamide; N-(5-tetrazolyl)-7-amino-8-ethoxy-4-oxo-4H-pyrimido[2,1-b]benzothiazole-3-carboxamide; N-(5-tetrazolyl)-7-amino-8-hydroxy-4-oxo-4H-pyrimido[2,1-b]benzothiazole-3-carboxamide; N-(5-tetrazolyl)-7-amino-8-chloro-4-oxo-4H-pyrimido[2,1-b]benzothiazole-3-carboxamide; and N-(5-tetrazolyl)-7-amino-8-fluoro-4-oxo-4H-pyrimido[2,1-b]benzothiazole-3-carboxamide.

Sources & evidence

ORD record
ord-4c8654d646514b8b8c68a61b0ed0f007
Source dataset
uspto-grants-1977_08
Patent number
US04041163

Reaction notes

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