3-(4-Fluoro-phenyl)-benzofuran-6-ol → (2S)-3-(4-{3-[3-(4-Fluoro-phenyl)-benzofuran-6-yloxy]-prop-1-ynyl}-phenyl)-2-methoxy-propionic acid

Participants

Reaction Steps

The title compound was prepared from (2S)-3-[4-(3-Chloro-prop-1-ynyl)-phenyl]-2-methoxy-propionic acid ethyl ester from Example 5, Step A and 6-hydroxy-3-(4-fluorophenyl)benzofurane in a manner analogous to that described for Example 5, Step B. MS(ES) for C27H21FO5 [M−H]−: 443.2.

Provenance & Evidence