Morpholine → HCID 70632586, compound

HRID 462270Notes

Reaction equation

[S:1]1[CH:5]=[CH:4][CH:3]=[C:2]1[CH2:6][C:7]([NH:9][CH:10]1[C:39](=[O:40])[N:12]2[C:13]([C:23]([O:25][CH:26]([C:33]3[CH:38]=[CH:37][CH:36]=[CH:35][CH:34]=3)[C:27]3[CH:32]=[CH:31][CH:30]=[CH:29][CH:28]=3)=[O:24])=[C:14]([N:17]3[CH2:22][CH2:21]O[CH2:19][CH2:18]3)[CH2:15][S:16][C@H:11]12)=[O:8].N1CCOC[CH2:42]1>>[S:1]1[CH:5]=[CH:4][CH:3]=[C:2]1[CH2:6][C:7]([NH:9][CH:10]1[C:39](=[O:40])[N:12]2[C:13]([C:23]([O:25][CH:26]([C:27]3[CH:28]=[CH:29][CH:30]=[CH:31][CH:32]=3)[C:33]3[CH:38]=[CH:37][CH:36]=[CH:35][CH:34]=3)=[O:24])=[C:14]([N:17]3[CH2:18][CH2:19][CH2:42][CH2:21][CH2:22]3)[CH2:15][S:16][C@H:11]12)=[O:8]

Participants

Reactant 2

HCID 8083Morpholine

HCID 70632798HCID 70632798, compound

Product 1

HCID 70632586HCID 70632586, compound

Procedure

By employing the procedures and starting material of Example 2 and substituting piperidine for morpholine the title compound was prepared.

Sources & evidence

ORD record: ord-06d1726eae3f44cb852da42279bd3456
Source dataset: uspto-grants-1977_12
DOI: 10.6084/m9.figshare.5104873.v1
Patent number: US04065621

Reaction notes

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