1-(4-Bromophenyl)-4-methylpiperazine → [5-(3-Methanesulfonyl-phenyl)-[1,2,4]triazolo[1,5-a]pyridin-2-yl]-[4-(4-methyl-piperazin-1-yl)-phenyl]-amine

Participants

Role	Name	HCID	Charge
Reactant	1-(4-Bromophenyl)-4-methylpiperazine	HCID 11817675	—
Reactant	5-(3-(Methylsulfonyl)phenyl)-[1,2,4]triazolo[1,5-a]pyridin-2-amine	HCID 59186437	—
Product	[5-(3-Methanesulfonyl-phenyl)-[1,2,4]triazolo[1,5-a]pyridin-2-yl]-[4-(4-methyl-piperazin-1-yl)-phenyl]-amine	HCID 59186482	—

Reaction Steps

[5-(3-Methanesulfonyl-phenyl)-[1,2,4]triazolo[1,5-a]pyridin-2-yl]-[4-(4-methyl-piperazin-1-yl)-phenyl]-amine was prepared from 5-(3-methanesulfonyl-phenyl)-[1,2,4]triazolo[1,5-a]pyridin-2-ylamine (75 mg, 0.26 mmol) and 1-(4-bromo-phenyl)-4-methyl-piperazine (73 mg, 0.28 mmol) in a manner analogous to Example 77 to yield [5-(3-methanesulfonyl-phenyl)-[1,2,4]triazolo[1,5-a]pyridin-2-yl]-[4-(4-methyl-piperazin-1-yl)-phenyl]-amine

Provenance & Evidence

DOI	10.6084/m9.figshare.5104873.v1
Patent number	US08633173B2
Source dataset	uspto-grants-2014_01
ORD ID	ord-7e9b2e21264c4d259712fcce62b9d313
Source note	uspto-grants-2014_01