HuagongsheHuagongshe Chemistry Print Report · For research reference only
1-(4-Fluorophenyl)pyrazole-4-boronic acid → [1-(4-fluoro-phenyl)1H-pyrazol-4-yl]-[1,2,4]triazolo[1,5-a]pyridine
Participants
| Role | Name | HCID | Charge |
|---|---|---|---|
| Reactant | 1-(4-Fluorophenyl)pyrazole-4-boronic acid | HCID 46738684 | — |
| Reactant | 8-Bromo-2-chloro-[1,2,4]triazolo[1,5-a]pyridine | HCID 67481370 | — |
| Product | [1-(4-fluoro-phenyl)1H-pyrazol-4-yl]-[1,2,4]triazolo[1,5-a]pyridine | HCID 86648363 | — |
Reaction Steps
2-Chloro-8-([1-(4-fluoro-phenyl)1H-pyrazol-4-yl]-[1,2,4]triazolo[1,5-a]pyridine was prepared from 8-bromo-2-chloro-[1,2,4]triazolo[1,5-a]pyridine and 1-(4-fluorophenyl)pyrazole-4-boronic acid in a manner analogous to Example 2c (0.45 g, 67%).
Provenance & Evidence
| DOI | 10.6084/m9.figshare.5104873.v1 |
|---|---|
| Patent number | US08633173B2 |
| Source dataset | uspto-grants-2014_01 |
| ORD ID | ord-165ce9346f0f487e81a91cf5f4cc56dc |
| Source note | uspto-grants-2014_01 |