2-(4-Pyridinyl)cyclopropanecarboxylic acid → HCID 58349682, compound

HRID 476274Notes

Reaction equation

HRID 476274 reaction equation
[N:1]1[CH:6]=[CH:5][C:4]([CH:7]2[CH2:9][CH:8]2[C:10]([OH:12])=O)=[CH:3][CH:2]=1.[CH3:13][NH:14][C@H:15]1[CH2:34][N:19]2[C:20]3[C:25]([C:26]([CH2:27][C:28]([O:30]CCC)=[O:29])=[C:18]2[CH2:17][CH2:16]1)=[CH:24][CH:23]=[CH:22][CH:21]=3>>[CH3:13][N:14]([C:10]([CH:8]1[CH2:9][CH:7]1[C:4]1[CH:3]=[CH:2][N:1]=[CH:6][CH:5]=1)=[O:12])[C@H:15]1[CH2:34][N:19]2[C:20]3[C:25]([C:26]([CH2:27][C:28]([OH:30])=[O:29])=[C:18]2[CH2:17][CH2:16]1)=[CH:24][CH:23]=[CH:22][CH:21]=3

Participants

3

Reactant 2

HCID 438102852-(4-Pyridinyl)cyclopropanecarboxylic acidHCID 86655417propyl [(7R)-7-(methylamino)-6,7,8,9-tetrahydropyrido[1,2-a]indol-10-yl]acetate

Product 1

HCID 58349682HCID 58349682, compound

Procedure

The title compound was prepared using analogous procedures described in Example 1 (Method A) from 2-(pyridin-4-yl)cyclopropanecarboxylic acid and propyl [(7R)-7-(methylamino)-6,7,8,9-tetrahydropyrido[1,2-a]indol-10-yl]acetate. MS (+ESI) m/z: 404.

Sources & evidence

ORD record
ord-192aa3660f424c88a423a6e14d1f9def
Source dataset
uspto-grants-2014_01
Patent number
US08637671B2

Reaction notes

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