3-(Piperidine-1-sulfonyl)benzoic acid → HCID 58349692, compound

HRID 476283Notes

Reaction equation

HRID 476283 reaction equation
[N:1]1([S:7]([C:10]2[CH:11]=[C:12]([CH:16]=[CH:17][CH:18]=2)[C:13]([OH:15])=O)(=[O:9])=[O:8])[CH2:6][CH2:5][CH2:4][CH2:3][CH2:2]1.[CH3:19][NH:20][C@H:21]1[CH2:40][N:25]2[C:26]3[C:31]([C:32]([CH2:33][C:34]([O:36]CCC)=[O:35])=[C:24]2[CH2:23][CH2:22]1)=[CH:30][CH:29]=[CH:28][CH:27]=3>>[CH3:19][N:20]([C:13](=[O:15])[C:12]1[CH:16]=[CH:17][CH:18]=[C:10]([S:7]([N:1]2[CH2:2][CH2:3][CH2:4][CH2:5][CH2:6]2)(=[O:8])=[O:9])[CH:11]=1)[C@H:21]1[CH2:40][N:25]2[C:26]3[C:31]([C:32]([CH2:33][C:34]([OH:36])=[O:35])=[C:24]2[CH2:23][CH2:22]1)=[CH:30][CH:29]=[CH:28][CH:27]=3

Participants

3

Reactant 2

HCID 7678893-(Piperidine-1-sulfonyl)benzoic acidHCID 86655417propyl [(7R)-7-(methylamino)-6,7,8,9-tetrahydropyrido[1,2-a]indol-10-yl]acetate

Product 1

HCID 58349692HCID 58349692, compound

Procedure

The title compound was prepared using analogous procedures described in Example 1 (Method A) from 3-(piperidin-1-ylsulfonyl)benzoic acid and propyl [(7R)-7-(methylamino)-6,7,8,9-tetrahydropyrido[1,2-a]indol-10-yl]acetate. MS (+ESI) m/z: 510.

Sources & evidence

ORD record
ord-7bbd2f568c0e472d999d01a54d5b7aef
Source dataset
uspto-grants-2014_01
Patent number
US08637671B2

Reaction notes

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