2,6-Dimethyl-8-ethyl-1-deazapurine → HCID 86752959, compound

HRID 481399Notes

Reaction equation

HRID 481399 reaction equation
[CH2:1]([O:3][C:4]([C:6]1([C:12]2[S:13][C:14]([CH2:17]Cl)=[CH:15][CH:16]=2)[CH2:11][CH2:10][O:9][CH2:8][CH2:7]1)=[O:5])[CH3:2].[CH2:19]([C:21]1[NH:22][C:23]2[C:24]([N:31]=1)=[N:25][C:26]([CH3:30])=[CH:27][C:28]=2[CH3:29])[CH3:20]>>[CH2:1]([O:3][C:4]([C:6]1([C:12]2[S:13][C:14]([CH2:17][N:31]3[C:24]4=[N:25][C:26]([CH3:30])=[CH:27][C:28]([CH3:29])=[C:23]4[N:22]=[C:21]3[CH2:19][CH3:20])=[CH:15][CH:16]=2)[CH2:11][CH2:10][O:9][CH2:8][CH2:7]1)=[O:5])[CH3:2]

Participants

3

Reactant 2

HCID 98153742,6-Dimethyl-8-ethyl-1-deazapurineHCID 57224386HCID 57224386, compound2×

Product 1

HCID 86752959HCID 86752959, compound

Procedure

The product of Step 4, above (40), was alkylated as described in Example 1, Step 5, using 2-ethyl-5,7-dimethylimidazo[4,5-b]pyridine (7) to obtain the title compound (41).

Sources & evidence

ORD record
ord-9d0b6b5931b544cdac2491eb3cdee883
Source dataset
uspto-grants-1998_08
Patent number
US05789415

Reaction notes

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