5-Chloroindole → 5-chloro-3-(1,2,3,6-tetrahydropyridin-4-yl)-1H-indole

Beteiligte Stoffe

Reaktionsschritte

The title compound was prepared in a fashion similar to that described in Preparation 30 from 5-chloroindole (3.0 g, 20 mmol) and 4-piperidone hydrochloride hydrate (6.0 g, 40 mmol). The product was isolated as a yellow solid. Yield 1.45 g (31%). mp 185°-188° C. FDMS m/e=234 (M+ of free base).

Herkunft & Nachweise