(Pyridin-4-yl)boronic acid → 2-(4-Pyridyl)furan-4-carboxylic acid

HRID 494185Notes

Reaction equation

HRID 494185 reaction equation
Br[C:2]1[O:3][CH:4]=[C:5]([C:7]([OH:9])=[O:8])[CH:6]=1.[N:10]1[CH:15]=[CH:14][C:13](B(O)O)=[CH:12][CH:11]=1>>[N:10]1[CH:15]=[CH:14][C:13]([C:2]2[O:3][CH:4]=[C:5]([C:7]([OH:9])=[O:8])[CH:6]=2)=[CH:12][CH:11]=1

Participants

3

Reactant 2

HCID 2734379(Pyridin-4-yl)boronic acidHCID 133335605-Bromofuran-3-carboxylic acid

Product 1

HCID 689464382-(4-Pyridyl)furan-4-carboxylic acid

Procedure

Using the procedure outlined in Description 29, the title compound was prepared from 2-bromo-furan-4-carboxylic acid (S. W. En, M. C. Yuen, H. N. C. Wong, Tetrahedron, 1996, 52(37), 12137) and 4-pyridylboronic acid.

Sources & evidence

ORD record
ord-4d70875c53104dc9b9a347e9de94e56c
Source dataset
uspto-grants-2009_05
Patent number
US07538121B2

Reaction notes

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