Pyridine sulfonamide → 2-{4-[6-chloro-2-ethyl-5-(trifluoromethyl)-1H-benzimidazol-1-yl]phenyl}ethyl 2-pyridinylsulfonylcarbamate

Participants

Role	Name	HCID	Charge
Reactant	Pyridine sulfonamide	HCID 12000791	—
Reactant	2-{4-[6-chloro-2-ethyl-5-(trifluoromethyl)-1H-benzimidazol-1-yl]phenyl}ethyl 3-pyridinylsulfonylcarbamate	HCID 21875896	—
Product	2-{4-[6-chloro-2-ethyl-5-(trifluoromethyl)-1H-benzimidazol-1-yl]phenyl}ethyl 2-pyridinylsulfonylcarbamate	HCID 21876180	—

Reaction Steps

The title compound was prepared according to the procedure described in step 2 of Example 243 from 2-pyridinesulfonamide (Naito, T.; et al., Chem. Pharm. Bull., 1955, 3, 38) and 2-[4-(2-ethyl-5,7-dimethyl-3H-imidazo[4,5-b]pyridin-3-yl)phenyl]ethylcarbamate (step 1 of Example 243).

Provenance & Evidence

DOI	10.6084/m9.figshare.5104873.v1
Patent number	US06710054B2
Source dataset	uspto-grants-2004_03
ORD ID	ord-ef7998a4244b4be9976af6216d86b046
Source note	uspto-grants-2004_03