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HuagongsheHuagongshe Chemistry Print Report · For research reference only
HRID 511410Generated: November 1, 2026

HCID 67255163, compound → HCID 58292971, compound

https://huagongshe.com/reaction/511410

Reaction equation

Participants

RoleNameHCIDCharge
ReactantHCID 67255163HCID 67255163—
ReactantDiethyl (4-{[4-chloro-5-(trifluoromethyl)pyrimidin-2-yl]amino}benzyl)phosphonateHCID 86654003—
ProductHCID 58292971HCID 58292971—

Reaction Steps

The title product was prepared according to the procedure for Example 102 using diethyl (4-{[4-chloro-5-(trifluoromethyl)pyrimidin-2-yl]amino}benzyl)phosphonate and 7-amino-2-methyl-4-(2H-tetrazol-5-yl)-2,3-dihydro-1H-isoindol-1-one (Compound 181A). MS (ES+): m/z 618.33 (100) [MH+]; HPLC: tR=1.13 min (UPLC, purity).

Provenance & Evidence

DOI10.6084/m9.figshare.5104873.v1
Patent numberUS09096624B2
Source datasetuspto-grants-2015_08
ORD IDord-940c95907d1c4f7fa0c6d752dca83563
Source noteuspto-grants-2015_08