HCID 90030461, compound → HCID 90030909, compound

Participants

Reaction Steps

Using similar reaction conditions as described in step-ii of example-7, tert-butyl 4-(6-(3-(1-(3-fluorobenzyl)-1H-pyrazol-4-yl)-1-tosyl-1H-pyrrolo[2,3-b]pyridin-5-yl)pyridin-3-yl)piperazine-1-carboxylate (800 mg, 1.130 mmol) was deprotected in TFA/DCM (3/10 ml) to afford 600 mg (87.4% yield) of the titled compound. MS: m/z=608.2 (M+1).

Provenance & Evidence