HCID 90031293, compound → HCID 118524115, compound

Participants

Reaction Steps

Using similar reaction conditions as described in step-ii of example-7, tert-butyl 4-(3-fluoro-5-(3-(1-(3-fluorobenzyl)-1H-pyrazol-4-yl)-1-tosyl-1H-pyrrolo[2,3-b]pyridin-5-yl)pyridin-2-yl)piperazine-1-carboxylate (step 1 product of example 173) (550 mg, 0.758 mmol) was deprotected in methanol/HCl in dioxane (5/5 ml) to afford 342 mg (72% yield) of the titled compound. MS: m/z=626.5 (M+1).

Provenance & Evidence