4-[(Methylsulfonyl)methyl]phenylboronic acid → 4-[5-(4-Methanesulfonylmethylphenyl)-2,3-dihydrofuro[2,3-c]pyridin-2-yl]-piperidine-1-carboxylic acid tert-butyl ester

Participants

Reaction Steps

The title compound is prepared from 4-(5-chloro-2,3-dihydro-furo[2,3-c]pyridin-2-yl)-piperidine-1-carboxylic acid tert-butyl ester and 4-(methanesulfonylmethyl)phenyl boronic acid following a procedure analogous to that described for Intermediate 10. LC (method 1): tR=1.55 min; Mass spectrum (ESI+): m/z=473 [M+H]+.

Provenance & Evidence