Morpholine → HCID 67157674, compound

Participants

Reaction Steps

As described for example 59, 6-[3-(4-fluoro-phenyl)-5-methyl-isoxazol-4-ylmethoxy]-pyridazine-3-carboxylic acid ethyl ester (143 mg, 0.4 mmol) was converted, using morpholine instead of aminomethylcyclopropane, to the title compound (132 mg, 83%) which was obtained as a light yellow solid. MS: m/e=399.1 [M+H]+.

Provenance & Evidence