7-Isopropoxy-1H-indole → 7-Isopropoxy-2-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-indole

HRID 550153Notes

Reaction equation

HRID 550153 reaction equation
Cl[C:2]1[CH:3]=[CH:4][CH:5]=[C:6]2[C:10]=1[NH:9][C:8]([B:11]1[O:15][C:14]([CH3:17])([CH3:16])[C:13]([CH3:19])([CH3:18])[O:12]1)=[CH:7]2.[CH:20]([O:23]C1C=CC=C2C=1NC=C2)([CH3:22])[CH3:21]>>[CH:20]([O:23][C:2]1[CH:3]=[CH:4][CH:5]=[C:6]2[C:10]=1[NH:9][C:8]([B:11]1[O:15][C:14]([CH3:17])([CH3:16])[C:13]([CH3:19])([CH3:18])[O:12]1)=[CH:7]2)([CH3:22])[CH3:21]

Participants

3

Reactant 2

HCID 219401147-Isopropoxy-1H-indoleHCID 532172117-Chloro-2-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-YL)-1H-indole

Product 1

HCID 591331207-Isopropoxy-2-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-indole

Procedure

Prepared according to a procedure analogous to that described for 7-chloro-2-(4,4,5,5-tetramethyl[1,3,2]dioxaborolan-2-yl)-1H-indole using 7-isopropoxy-1H-indole.

Workup

  1. customPrepared

Sources & evidence

ORD record
ord-fde46cb8d2064f6bb5d5e5f887dd54b4
Source dataset
uspto-grants-2011_05
Patent number
US07943767B2

Reaction notes

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