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HuagongsheHuagongshe Chemistry Print Report · For research reference only
HRID 550717Generated: October 30, 2026

(3-Acetamidophenyl)boronic acid → Fen1-IN-5

https://huagongshe.com/reaction/550717

Reaction equation

Participants

RoleNameHCIDCharge
Reactant(3-Acetamidophenyl)boronic acidHCID 157274—
Reactant1-(3-Bromo-benzyl)-3-hydroxy-1H-thieno[3,2-d]pyrimidine-2,4-dioneHCID 11544874—
ProductFen1-IN-5HCID 11611180—

Reaction Steps

The title compound was prepared from 1-(3-Bromo-benzyl)-3-hydroxy-1H-thieno[3,2-d]pyrimidine-2,4-dione (from previous example) and 3-acetamino-phenyl boronic acid via general procedure C. The crude product was purified by mass-triggered preparative HPLC.

Provenance & Evidence

DOI10.6084/m9.figshare.5104873.v1
Patent numberUS07947691B2
Source datasetuspto-grants-2011_05
ORD IDord-86c34690e4c344d99def78d418731183
Source noteuspto-grants-2011_05