Dimethylsulphamoyl chloride → HCID 66998736, compound

HRID 559262Notes

Reaction equation

[Cl:1][C:2]1[CH:7]=[C:6]([Cl:8])[CH:5]=[CH:4][C:3]=1[C:9]1[C:27](=[O:28])[N:26]([CH3:29])[C:12]2[N:13]([CH3:25])[C:14]3[C:19]([C:11]=2[CH:10]=1)=[CH:18][C:17]([C:20]1[NH:21][N:22]=[CH:23][CH:24]=1)=[CH:16][CH:15]=3.[CH3:30][N:31]([CH3:36])[S:32](Cl)(=[O:34])=[O:33]>>[CH3:30][N:31]([CH3:36])[S:32]([N:22]1[CH:23]=[CH:24][C:20]([C:17]2[CH:18]=[C:19]3[C:14](=[CH:15][CH:16]=2)[N:13]([CH3:25])[C:12]2[N:26]([CH3:29])[C:27](=[O:28])[C:9]([C:3]4[CH:4]=[CH:5][C:6]([Cl:8])=[CH:7][C:2]=4[Cl:1])=[CH:10][C:11]3=2)=[N:21]1)(=[O:34])=[O:33]

Participants

Reactant 2

HCID 83372Dimethylsulphamoyl chloride

HCID 16226262HCID 16226262, compound

Product 1

HCID 66998736HCID 66998736, compound

Procedure

The process is carried out as indicated in Example 99 above, with the compound from Example 39, 3-(2,4-dichlorophenyl)-1,9-dimethyl-6-(2H-pyrazol-3-yl)-1,9-dihydropyrido[2,3-b]indol-2-one, and dimethyl sulphamoyl chloride.

Sources & evidence

ORD record: ord-0bfd7f563f594010a1d0b1b0140b6196
Source dataset: uspto-grants-2011_11
DOI: 10.6084/m9.figshare.5104873.v1
Patent number: US08063061B2

Reaction notes

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