4-Methoxycinnamic Acid → HCID 67005100, Verbindung

Beteiligte Stoffe

Reaktionsschritte

Acylation of 1-(4-benzyl-piperazin-1-yl)-(S)-2-(4-pentyl-benzylamino)-3-phenyl-propan-1-one (43.5 mg, 0.09 mmol) according to the procedure described for the preparation of Example 1 with trans-4-methoxy-cinnamic acid (17.6 mg, 0.099 mmol) gave 27.7 mg (48%) of N—[(S)-1-benzyl-2-(4-benzyl-piperazin-1-yl)-2-oxo-ethyl]-3-(4-methoxy-phenyl)-N-(4-pentyl-benzyl)-acrylamide. LC-MS: tR=1.00 min; [M+H]+=644.50.

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