Ethyl-[2-(4,4,5,5-tetramethyl-[1,3,2]dioxaborolan-2-yl)-5-trifluoromethylbenzyl]-carbamic acid benzyl ester → {2'-[(Benzyloxycarbonyl-ethyl-amino)-methyl]-4,4'-bis-trifluoromethyl-biphenyl-3-yl}-acetic acid ethyl ester

Participants

Reaction Steps

Prepared according to the procedure described in Example 1, Step 4, using the following starting materials: ethyl-[2-(4,4,5,5-tetramethyl-[1,3,2]dioxaborolan-2-yl)-5-trifluoromethyl-benzyl]-carbamic acid benzyl ester and (5-trifluoromethanesulfonyloxy-2-trifluoromethyl-phenyl)-acetic acid ethyl ester.

Provenance & Evidence