HuagongsheHuagongshe Chemistry Print Report · For research reference only
HCID 58221469, compound → HCID 86693249, compound
Participants
| Role | Name | HCID | Charge |
|---|---|---|---|
| Reactant | HCID 58221469 | HCID 58221469 | — |
| Reactant | 9-Bromo-8-fluoro-4,5-dihydro-[1]benzoxepino[5,4-d]thiazole-2-carboxamide | HCID 86693059 | — |
| Product | HCID 86693249 | HCID 86693249 | 9% |
Reaction Steps
Similar to as described in General Procedure G, 9-bromo-8-fluoro-4,5-dihydrobenzo[2,3]oxepino[4,5-d]thiazole-2-carboxamide was reacted with 2-(1-methyl-1H-imidazol-4-yl)but-3-yn-2-ol (WO2009/158011 A1) to give the titled compound as colorless solid (19 mg, 9%).
Provenance & Evidence
| DOI | 10.6084/m9.figshare.5104873.v1 |
|---|---|
| Patent number | US09034866B2 |
| Source dataset | uspto-grants-2015_05 |
| ORD ID | ord-77cf9c69ce764675a3c923dfdfdfe758 |
| Source note | uspto-grants-2015_05 |