HCID 178466095, compound → HCID 178466070, compound

HRID 57801Notes

Reaction equation

HRID 57801 reaction equation
C([O:3][C:4](=[O:25])[CH2:5][C:6]1[C:11](=[O:12])[N:10]2[N:13]=[C:14]([C:16]3[CH:21]=[CH:20][C:19]([O:22][CH2:23][CH3:24])=[CH:18][CH:17]=3)[CH:15]=[C:9]2[NH:8][CH:7]=1)C.C(OC1C=CC(C2C=C(N)NN=2)=CC=1)C>>[CH2:23]([O:22][C:19]1[CH:18]=[CH:17][C:16]([C:14]2[CH:15]=[C:9]3[NH:8][CH:7]=[C:6]([CH2:5][C:4]([OH:25])=[O:3])[C:11](=[O:12])[N:10]3[N:13]=2)=[CH:21][CH:20]=1)[CH3:24]

Participants

3

Reactant 2

HCID 178466095HCID 178466095, compoundHCID 178470742HCID 178470742, compound

Product 1

HCID 178466070HCID 178466070, compound

Procedure

The expected compound was obtained according to general procedure G using [2-(4-ethoxy-phenyl)-7-oxo-4,7-dihydro-pyrazolo[1,5-a]pyrimidin-6-yl]acetic acid ethyl ester. The starting material was obtained according to general procedure E using 5-(4-ethoxy-phenyl)-2H-pyrazol-3-ylamine. The expected compound was isolated as white powder.

Workup

  1. customThe starting material was obtained

Sources & evidence

ORD record
ord-e98ea91ba14a4e75bdc67eeca88f3662
Source dataset
uspto-grants-2016_09
Patent number
US09434745B2

Reaction notes

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