Furan-3-boronic acid → HCID 54211699, compound

HRID 581942Notes

Reaction equation

HRID 581942 reaction equation
F.[NH2:2][C:3]1[N:8]=[CH:7][C:6]([C:9]2[CH:10]=[C:11]([NH:15][C:16]3[CH:21]=[CH:20][C:19](I)=[CH:18][C:17]=3[N+:23]([O-:25])=[O:24])[CH:12]=[CH:13][CH:14]=2)=[CH:5][N:4]=1.[O:26]1[CH:30]=[CH:29][C:28](B(O)O)=[CH:27]1>>[NH2:2][C:3]1[N:8]=[CH:7][C:6]([C:9]2[CH:10]=[C:11]([NH:15][C:16]3[CH:21]=[CH:20][C:19]([C:28]4[CH:29]=[CH:30][O:26][CH:27]=4)=[CH:18][C:17]=3[N+:23]([O-:25])=[O:24])[CH:12]=[CH:13][CH:14]=2)=[CH:5][N:4]=1

Participants

3

Reactant 2

HCID 2734358Furan-3-boronic acidHCID 67482348HCID 67482348, compound

Product 1

HCID 54211699HCID 54211699, compound

Procedure

N-(3-(2-Aminopyrimid-5-yl)phenyl)-4-(3-furanyl)-2-nitroaniline (71) was prepared analogously from 6l (Example 10) and 3-furanylboronic acid in quantitative yield. Mp 185-186° C.

Sources & evidence

ORD record
ord-829d66a7d0e3467d8de803c1830501a4
Source dataset
uspto-grants-1999_07
Patent number
US05922724

Reaction notes

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