2,2,2-Trifluoroethyl trifluoromethanesulfonate → HCID 54381097, compound

HRID 582078Notes

Reaction equation

HRID 582078 reaction equation
FC(F)(F)S(O[CH2:7][C:8]([F:11])([F:10])[F:9])(=O)=O.[NH:14]1[C:18]2[CH:19]=[CH:20][CH:21]=[CH:22][C:17]=2[N:16]=[C:15]1[NH:23][CH:24]1[CH2:29][CH2:28][N:27](C(OCC)=O)[CH2:26][CH2:25]1>>[F:9][C:8]([F:11])([F:10])[CH2:7][N:14]1[C:18]2[CH:19]=[CH:20][CH:21]=[CH:22][C:17]=2[N:16]=[C:15]1[NH:23][CH:24]1[CH2:29][CH2:28][NH:27][CH2:26][CH2:25]1

Participants

3

Reactant 2

HCID 803662,2,2-Trifluoroethyl trifluoromethanesulfonateHCID 30184551-Piperidinecarboxylic acid, 4-(1H-benzimidazol-2-ylamino)-, ethyl ester

Product 1

HCID 54381097HCID 54381097, compound

Procedure

Prepare by the method of Preparation 14 using 2,2,2-trifluoroethyl trifluoromethanesulfonate and (1H-benzimidazol-2-yl)(1-ethoxycarbonylpiperidin-4-yl)amine to give the title compound.

Sources & evidence

ORD record
ord-ebd692cc96804fc7bc1a77527cd006d8
Source dataset
uspto-grants-1999_07
Patent number
US05922737

Reaction notes

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