N-(1,2,3,4-tetrahydro-quinolin-6-yl)acetamide → N-[1-[1-(3,4-Dimethoxybenzoyl)-2-methyl-1,2,3,4-tetrahydroquinolin-4-yl]-1,2,3,4-tetrahydroquinolin-6-yl]acetamide

참여 물질

반응 단계

Starting with cis-1-(3,4-dimethoxybenzoyl)-2-methyl-1,2,3,4-tetrahydro-4-quinolinol (350 mg, 1.07 mmol) prepared in Reference Example 1 and N-(1,2,3,4-tetrahydro-quinolin-6-yl)acetamide (475 mg, 2.50 mmol), the same procedure as shown in Example 1 was repeated to give the titled compound (38 mg, yield: 7%) as a colorless oil. (cis:trans=1:1.7)

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