2-(3-Aminophenyl)ethanesulfonamide → (R)-3-[(4-(2-(Phenoxymethyl)pyrrolidin-1-yl)-1,3,5-triazin-2-yl)amino]-benzenemethanesulfonamide

Beteiligte Stoffe

Rolle	Name	HCID	Einwaage
Edukt	2-(3-Aminophenyl)ethanesulfonamide	HCID 58236871	—
Edukt	rac-3-[(4-(2-Methoxymethylpiperidin-1-yl)-1,3,5-triazin-2-yl)amino]-benzenemethanesulfonamide	HCID 60197106	—
Edukt	3-[(4-Chloro-1,3,5-triazin-2-yl)amino]benzenemethanesulfonamide	HCID 86679822	—
Produkt	(R)-3-[(4-(2-(Phenoxymethyl)pyrrolidin-1-yl)-1,3,5-triazin-2-yl)amino]-benzenemethanesulfonamide	HCID 60197500	—

Reaktionsschritte

B28 was prepared following the procedure reported for B4 using the intermediates A1 and A3. It was obtained as a white crystalline powder; yield: 140 mg (35%). MS (ES) C21H24N6O3S requires: 440. found: 441 (M+H)+.

Herkunft & Nachweise

DOI	10.6084/m9.figshare.5104873.v1
Patentnummer	US09226929B2
Quelldatensatz	uspto-grants-2016_01
ORD ID	ord-3ed22f00b73a4e39831cde877448d539
Quellennotiz	uspto-grants-2016_01