(3-Carbamoylphenyl)boronic acid → HCID 178513632, compound

Participants

Reaction Steps

The product was prepared according to General Procedure 3, described in Example 22, starting from 5-bromo-N-[3-(1H-tetrazol-5-yl)phenyl]thiophene-2-sulfonamide (Intermediate 17) (19 mg, 0.05 mmol) and 3-aminocarbonylphenylboronic acid (10 mg, 0.06 mmol) giving 2.7 mg (13%) of the title compound. MS (ESI+) calcd for C18H14N6O3S2 426.056880, found 426.057610.

Provenance & Evidence