(2-Chloropyrimidin-5-yl)boronic acid → HCID 131735235, compound

HRID 626953Notes

Reaction equation

HRID 626953 reaction equation
[CH:1]12[CH2:10][CH2:9][CH:5]([NH:6][C:7]1=[O:8])[CH2:4][NH:3][CH2:2]2.Cl[C:12]1[N:17]=[CH:16][C:15]([B:18]([OH:20])[OH:19])=[CH:14][N:13]=1>>[O:8]=[C:7]1[CH:1]2[CH2:10][CH2:9][CH:5]([CH2:4][N:3]([C:12]3[N:17]=[CH:16][C:15]([B:18]([OH:20])[OH:19])=[CH:14][N:13]=3)[CH2:2]2)[NH:6]1

Participants

3

Reactant 2

HCID 21747362(2-Chloropyrimidin-5-yl)boronic acidHCID 78149444HCID 78149444, compound

Product 1

HCID 131735235HCID 131735235, compound

Procedure

The title compound was prepared from 3,6-diazabicyclo[3.2.2]nonan-7-one and (2-chloropyrimidin-5-yl)boronic acid in accordance with General Method C.

Sources & evidence

ORD record
ord-6d988dd4681848578051c3ce8cd8572c
Source dataset
uspto-grants-2016_04
Patent number
US09309243B2

Reaction notes

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