HuagongsheHuagongshe Chemistry Print Report · For research reference only
(4-Methoxyphenyl)boronic acid → 6-Bromo-3-(4-methoxyphenyl)imidazo[1,2-a]pyridine
Participants
| Role | Name | HCID | Charge |
|---|---|---|---|
| Reactant | (4-Methoxyphenyl)boronic acid | HCID 201262 | — |
| Reactant | 6-Bromo-3-iodoimidazo(1,2-a)pyridine | HCID 22031632 | — |
| Product | 6-Bromo-3-(4-methoxyphenyl)imidazo[1,2-a]pyridine | HCID 22031458 | — |
Reaction Steps
The title compound, brown oil (0.47 g, 72%), MS (ISP) m/z=303.4 [(M+H)+], was prepared in accordance with the general method of intermediate E from commercially available 6-bromo-3-iodoimidazo[1,2-a]pyridine (0.7 g, 2.17 mmol) and commercially available 4-methoxy-phenylboronic acid (0.36 g, 2.38 mmol).
Provenance & Evidence
| DOI | 10.6084/m9.figshare.5104873.v1 |
|---|---|
| Patent number | US09315502B2 |
| Source dataset | uspto-grants-2016_04 |
| ORD ID | ord-26816ee90cd74a9b9ec0ff7a9ef7e678 |
| Source note | uspto-grants-2016_04 |