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HuagongsheHuagongshe Chemistry Print Report · For research reference only
HRID 629268Generated: October 27, 2026

(4-Methoxyphenyl)boronic acid → 6-Bromo-3-(4-methoxyphenyl)imidazo[1,2-a]pyridine

https://huagongshe.com/reaction/629268

Reaction equation

Participants

RoleNameHCIDCharge
Reactant(4-Methoxyphenyl)boronic acidHCID 201262—
Reactant6-Bromo-3-iodoimidazo(1,2-a)pyridineHCID 22031632—
Product6-Bromo-3-(4-methoxyphenyl)imidazo[1,2-a]pyridineHCID 22031458—

Reaction Steps

The title compound, brown oil (0.47 g, 72%), MS (ISP) m/z=303.4 [(M+H)+], was prepared in accordance with the general method of intermediate E from commercially available 6-bromo-3-iodoimidazo[1,2-a]pyridine (0.7 g, 2.17 mmol) and commercially available 4-methoxy-phenylboronic acid (0.36 g, 2.38 mmol).

Provenance & Evidence

DOI10.6084/m9.figshare.5104873.v1
Patent numberUS09315502B2
Source datasetuspto-grants-2016_04
ORD IDord-26816ee90cd74a9b9ec0ff7a9ef7e678
Source noteuspto-grants-2016_04